http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2007099962-A1

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filingDate 2004-12-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2007-05-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2007099962-A1
titleOfInvention 5,6-Dihydropyrin-2-one compounds useful as inhibitors of thrombin
abstract There is provided a compound of formula (I) wherein R 1 , R 2a , R 2b , R 3a , R 3b , R 4 , R 5 , R 6 , A, G and L have meanings given in the description, which compounds are useful as, or are useful as prodrugs of, competitive inhibitors of trypsin-like proteases, such as trombin, and thus, in particular, in the treatment of conditions where inhibition of thrombin is beneficial (e.g. conditions, such as thrombo-embolisms, where inhibition of trombin is required or desired, and/or conditions whereas anticoagulant therapy is indicated).
priorityDate 2003-12-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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Total number of triples: 1489.