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publicationDate 2006-06-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2006141043-A1
titleOfInvention Aqueous dispersion comprising stable nanoparticles of a water-insoluble thiazole derivative and excipients like middle chain triglycerides
abstract A process for the preparation of a stable dispersion of solid particles, in an aqueous medium comprising combining (a) a first solution comprising a substantially water-insoluble substance which is a thiazole compound of Formula I, a water-miscible organic solvent and an inhibitor with (b) an aqueous phase comprising water and optionally a stabiliser, thereby precipitating solid particles comprising the inhibitor and the substantially water-insoluble substance; and optionally removing the water-miscible organic solvent; wherein the inhibitor is a non-polymeric hydrophobic organic compound as defined in the description. n nAlso claimed are stable dispersions prepared by the process, solid particles prepared by the process and use of such particles.
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Total number of triples: 417.