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publicationDate 2006-06-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2006134087-A1
titleOfInvention ITI-D1 Kunitz domain mutants as hNE inhibitors
abstract Mutants of Kunitz domain 1 (ITI-D1) of human inter-alpha-trypsin inhibitor (ITI), are useful as inhibitors of human neutrophil elastase. Mutants characterized by one or more of the following substitutions (numbered to correspond to bovine pancreatic trypsin inhibitor, the archetypal Kunitz domain) are of particular interest: (a) Val15 or Ile15, (b) Ala16, (c) Phe18, (d) Pro19, (e) Arg1, (f) Pro2, and/or (g) Phe4.
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399382
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID436926
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID21788
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO97398
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5K2K7
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399383
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO97399
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP86242
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID8704
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID359833
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9DUE3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ65372
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP41359
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP62757
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID290257
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68921
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP62693
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP11211
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP78285
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID230996503
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9JGU1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP62756
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0GBX9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP11212
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458397476
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68920
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419571978
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP11187
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID449812109
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128479187
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID66629
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP09963
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ03332
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID449046755
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458397419
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID8467
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP00720
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9QSP4
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID25043
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5VKP2
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID422600743
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ86AA1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9QL89
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP03521
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP04365
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9QJT9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP27018
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP08311
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO01945
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP23916
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP14155
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0GBY4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8B0H4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB1AAA7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8B0H9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP00761
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID426049
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID57369551
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP00749
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0DOF3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP24304
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226406585
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ59149
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID20730
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP10646
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP11547
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP27359
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7Y2C0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ61955
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5RC19
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP24664
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http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID4922
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ00922
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Total number of triples: 408.