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filingDate 2003-10-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2006-01-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2006004024-A1
titleOfInvention Method for preparing risperidone
abstract Risperidone is prepared in a high yield by reacting 2,4-difluorophenyl(4-piperidinyl)methanone oxime hydrochloride and 3-(2-chloroethyl)-6,7,8,9-tetrahydro-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one in an aqueous alkali hydroxide solution having an alkali hydroxide concentration in the range of 20 to 40%.
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