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titleOfInvention Process for preparing acyclic HCV protease inhibitors
abstract Disclosed are highly convergent processes for preparing compounds of formula (I), which compounds are potent active agents for the treatment of hepatitis C virus (HCV) infection: n n n The disclosed processes use S N Ar-type coupling reactions between peptidic compounds having a hydroxyproline moiety of the following formula: n nand halogenated or sulfonated bromoquinoline compounds.
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Total number of triples: 456.