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publicationDate 2005-11-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2005245500-A1
titleOfInvention Beta-ketoamide compounds with MCH antagonistic activity
abstract Compounds of formula I n n nwherein the groups and residues A, B, b, X, Y, Z, R 1 , R 2 , R 3 , R 5a and R 5b have the meanings given in claim 1 . The invention further relates to pharmaceutical compositions containing at least one amide according to the invention. As a result of their MCH-receptor antagonistic activity the pharmaceutical compositions according to the invention are suitable for the treatment of metabolic disorders and/or eating disorders, particularly obesity, bulimia, anorexia, hyperphagia, and diabetes.
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Total number of triples: 2077.