http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2004171631-A1

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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-485
filingDate 2004-03-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5a387dd8921ceca41f59b7cd43eec035
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_44f6cb6e38b9754a09f9a018d2472a3d
publicationDate 2004-09-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2004171631-A1
titleOfInvention Orally administered analgesic compositions containing nalbuphine
abstract The present invention provides orally administered pharmaceutical compositions which contains an effective amount of free base or pharmaceutically acceptable salts of nalbuphine and/or nalbuphine ester, an oily substance, and a solubility-assisting agent. The oily substance is preferably sesame oil. The solubility-assisting agent is preferably benzyl benzoate. The pharmaceutical composition is useful as an analgesic. The compositions achieves a much higher bioavailability rate and yields much longer lasting effects on nalbuphine than other nalbuphine products currently in the market.
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