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filingDate 2001-09-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_33b7be11b6cf33b3dc8355617ea42bcd
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_63d4d918268e929da02cf4f942c411dd
publicationDate 2004-02-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2004029100-A1
titleOfInvention Rapid screen to identify p-glycoprotein substrates and high affinity modulators
abstract A novel method for identifying compounds that interact with P-glycoprotein that involves measuring the quenching of intrinsic tryptophan fluorescence is described. The method has many uses including (1) it can be used to screen drugs for their ability to interact with P-glycoprotein; (2) it can be used to screen for high affinity modulators of P-glycoprotein; and (3) it can be used to screen drugs that are potential hazards when used in combination with the modulators and (4) it can be used in methods of conducting target discovery/screening businesses.
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type http://data.epo.org/linked-data/def/patent/Publication

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