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publicationDate 2003-12-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2003232869-A1
titleOfInvention N3 alkylated benzimidazole derivatives as MEK inhibitors
abstract Disclosed are compounds of the formula I n n n and pharmaceutically acceptable salts and prodrugs thereof, wherein W, R 1 , R 2 , R 7 , R 8 , R 9 and R 10 are as defined in the specification. n Such compounds are MEK inhibitors and useful in the treatment of hyperproliferative diseases, such as cancer and inflammation, in mammals. Also disclosed is a method of using such compounds in the treatment of hyperproliferative diseases in mammals, and pharmaceutical compositions containing such compounds.
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Total number of triples: 2413.