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filingDate 2001-08-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2002-10-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2002160038-A1
titleOfInvention Liposomes containing oligonucleotides
abstract It is possible to radiosensitize tumor cells by administration of compositions containing the Human antisense c-raf- 1 oligodeoxyribonucleotide (ODN/oligo) sequence: 5 ′-GTGCTCCATTGATGC- 3 ′ (seq. # 1 ) wherein only the end bases are phosphorylated is a preferred embodiment. Antisense sequences of up to 40 bases which containing this sequence may be used in accord with the teachings of this disclosure. Compositions comprising a cationic liposome of dimethyldioctadecyl ammonium bromide, phosphatidylcholine and cholesterol may be used as a carrier system. The liposomes provide a new carrier system that is particularly useful for administration of sequences for therapy.
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