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filingDate 2000-12-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_38e500ba9dc5411d3a02f09ea5ed22f9
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_09638f19cf85c2013d6b06ca18651c90
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_e3a4934a3d95b1ac20ebfdf4d16593d1
publicationDate 2002-05-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2002052343-A1
titleOfInvention Salicylamides as serine protease inhibitors
abstract The present invention provides novel compounds of Formula I: n n n its prodrug forms, or pharmaceutically acceptable salts thereof. The compounds of this invention are inhibitors of serine proteases, Urokinase (uPA), Factor Xa (FXa), and/or Factor VIIa (FVIIa), and have utility as anti cancer agents and/or as anticoagulants for the treatment or prevention of thromboembolic disorders in mammals. The present invention also provides a process for the selective acylation of an amino group.
priorityDate 1999-12-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 699.