http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2002040018-A1

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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-4745
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-407
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-4745
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filingDate 2001-06-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_7c6cefc120ac0e54941c9710d6f30738
publicationDate 2002-04-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2002040018-A1
titleOfInvention Subtype selective melatonergics
abstract The invention relates to the use of MT 2 selective melatonergics as anticonvulsant agents and as analgesic agents. More specifically, the invention relates to the use of 6H-isoindolo[2,1-a]indoles or 5,6-dihydroindolo[2,1-a]isoquinolines as described herein which have melatonin agonist activity and which are selective for the MT 2 receptor as anticonvulsant agents or analgesic agents. The invention further relates to the use of 5,6-dihydroindolo[2,1-a]isoquinolines and 6,7-dihydro-5H-benzo[c]azepino[2,1-a]indoles as described herein which have melatonin antagonist activity and which are selective for the MT 2 receptor as pharmacological tools for delineation of physiological responses governed by MT 2 receptor activation either by melatonin or selective agonists disclosed herein and for treatment of disorders associated with overproduction of melatonin such as seasonal affective disorder (SAD) and shift work syndrome. Such melatonin antagonists are also useful for treating Parkinson's Disease.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2016077654-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-10555919-B2
priorityDate 2000-06-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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