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filingDate 2001-06-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_779be8e1126c4b4b0f483f0bc90a33db
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publicationDate 2002-02-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2002025957-A1
titleOfInvention Lactam inhibitors of factor Xa and method
abstract Lactam inhibitors are provided which have the structure n n n including pharmaceutically acceptable salts thereof and all stereoisomers thereof, and prodrug esters thereof, wherein n is 1 to 5; and n and R 1 , R 2 , R 3 , R 4 , R 5 , R 6 , R 7 , R 8 , R 9 , R 10 , R 10a , 10 11 and R 12 are as defined herein. These compounds are inhibitors of Factor Xa and thus are useful as anticoagulants. A method for treating cardiovascular diseases associated with thromboses is also provided.
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http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2009105322-A1
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priorityDate 2000-06-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID142309953
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID141983396
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID656606
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24391
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID136827
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID424114008
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2733832
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID406935663
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID141983438
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419506136
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID90721101
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID141983437
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID127717286
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5PJB2
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID142303989
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID141983440
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100301982
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419506158
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID18612618
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID141983434
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID91268869
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID142291669
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID432222851
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4449
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11194423
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10450
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO14595
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID90932114
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID432311771
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID91353511
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Total number of triples: 3216.