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filingDate 2021-04-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2022-07-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_453096e28f09ac2bb7cb78d84864bbde
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c52945f669ad340d5a05522a187990d0
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publicationDate 2022-07-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-11390629-B2
titleOfInvention 1,5-disubstituted 1,2,3-triazoles are inhibitors of Rac/Cdc42 GTPases
abstract Compounds are disclosed that inhibit RhoGTPases that are useful for inhibiting hyperproliferative and neoplastic diseases. Specifically, the compounds inhibit the GTPases Rac and Cdc42 that are overactive or overexpressed in signaling pathways in cancer and metastasis. Methods for treatment of cancer and hyperproliferative diseases are disclosed.
priorityDate 2016-04-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393971
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID53585
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID449097368
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393977
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6950218
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID8420
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID484513
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID432338778
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393981

Total number of triples: 637.