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filingDate 2019-07-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2022-06-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_241c6f9ae0d2e7b676abd990602b8760
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publicationDate 2022-06-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-11370742-B2
titleOfInvention Process and intermediates for the preparation of bilastine
abstract The invention relates to a process for preparing a compound of (III)whereinX is a leaving group; andR1 is C1-C6 alkyl;which comprises oxidative rearrangement of a compound of formula (II) or a solvate thereofCompounds of formula (III) are key intermediates in the synthesis of Bilastine.
priorityDate 2018-07-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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