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filingDate 2018-03-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2022-04-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_0d4ef1b5a35408d140b23bd1c36c0312
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publicationDate 2022-04-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-11304929-B2
titleOfInvention Tosylacetate based compounds and derivatives thereof as PHGDH inhibitors
abstract The present invention encompasses compounds of formula (I), wherein the groups R 1 to R, A 1 to A 4 and n have the meanings given in the claims and specification, their use as inhibitors of PHGDH, pharmaceutical compositions which contain compounds of this kind and their use as medicaments, especially as agents for treatment and/or prevention of oncological diseases.
priorityDate 2017-03-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID384983667
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID166935066
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8EWD1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ667X1
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID469793573
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA1WQP4
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID29255296
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1IS84
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID53628963
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID227112789
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID166935058
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID227113024
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP40510
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID166935059
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID14284
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2V9M1
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID469793561
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1J1W0
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID166935036
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ65T08
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP40054
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID150009356
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC3L181
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID11677
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP77962
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID155567512
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID155568226
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA1VYC2
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID166935047
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID280675
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ660S1
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135331313
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID155563606
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID166935048
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135331314
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID156122075
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID166935045
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA7ZPZ4
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID117916811
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2187
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID360149
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID166935046
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419587201
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC3LFJ0
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID7940935
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID166935044

Total number of triples: 3491.