http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-11267820-B2

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filingDate 2020-05-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2022-03-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_51141fd93fc883f1070ddd7e4cd23546
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_ee74d4b63e43b5c62af8dc1c6549229d
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publicationDate 2022-03-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-11267820-B2
titleOfInvention Tricyclic fused pyridin-2-one derivatives and their use as BRD4 inhibitors
abstract The present disclosure describes heterocyclic compounds of Formula I or, its stereoisomers, pharmaceutically acceptable salts, complexes, hydrates, solvates, tautomers, polymorphs, racemic mixtures, optically active forms and pharmaceutically active derivatives thereof and pharmaceutical compositions containing them as the active ingredient. The present disclosure also describes the synthesis and characterization of aforementioned compounds to exhibit high anticancer activity. The compounds of the present disclosure are useful as medicaments and their use in the manufacture of medicaments for treatment, prevention, or suppression of diseases, an conditions mediated b one or more BET family of bromodomains.
priorityDate 2015-09-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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Total number of triples: 421.