http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-11104703-B2

Outgoing Links

Predicate Object
assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_8cf2caf35a4f97a4534d8923f7fd25a4
classificationCPCAdditional http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K38-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/G01N2800-382
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/G01N2333-96433
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07K5-02
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K47-557
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07K5-0806
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07K5-1019
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07K7-02
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C12N9-99
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C12Q1-37
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/G01N33-573
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07K5-021
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K47-66
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P11-00
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07K5-02
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07K7-02
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K47-54
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C12Q1-37
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/G01N33-573
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P11-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K38-00
filingDate 2017-10-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2021-08-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_75ffa0520d0ab40a8c61c3dab4a20d84
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b0e38395cc23872f6ccbcae800fb4d16
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_e12dc9d52dfcdd67fa425ef134937356
publicationDate 2021-08-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-11104703-B2
titleOfInvention Binding compound and uses thereof
abstract Described are compounds for targeting proteases, e.g. serine proteases and their use in the diagnostic methods and methods for treatment of respiratory diseases such as cystic fibrosis. The compounds have the structure [H]—[B]-[A]; wherein [H] is a hydrophilic group, [B] is a subsite recognition group and [A] is a binding group; wherein A has the formula: —C(0)—CH 2 —NR 1 —COOR 2 and wherein [B] has the structure: (i) —[CO—CH 2 —NR 3 ]m-, or (ii) -[AA1-AA2]- or (iii) -(AA1-C0-CH 2 NR 3 )— or (iv) —(CO—CH 2 —NR 3 -AA1)- or (v) —(C0—CH 2 —NR 4 -AA1-AA3)-.
priorityDate 2016-10-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

Incoming Links

Predicate Subject
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2002156018-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2011024006-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2016118910-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-9929311-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-5550139-A
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-2470672-A1
isDiscussedBy http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID28983
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID21106254
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6301202
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID16613
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCF7EHU5
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457342965
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID493836
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID299606
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID199
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458396881
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID17393
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419523391
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID29260
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID676246
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCCAH72619
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO60109
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP83456
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9Y5Y6
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID489432
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3T478
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCV5NAL9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP19147
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP83348
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01012
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9TTN0
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16231
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID373926
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ16651
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO73860
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419505358
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ68Y56
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID414025332
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP22775
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP19104
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP70059
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP51588
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID454464170
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11990
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ28193
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9TSP2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO97399
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID566557
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO97398
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID4316
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16760442
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP22629
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP86348
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID47220
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID569750
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID107689
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID8371
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID397197
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419587903
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP23916
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID50701
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID395457
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP00634
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID418983
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID452705
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID451172592
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID18550
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6227
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP55032
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID21932394
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP35048
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID396495
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7311726
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458394834
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID54281
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID403850
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP35034
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP58727
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID396880
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID280828
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID424603604
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP35002
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID7099
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419586411
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID76560
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID452473801
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID6768
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID1476581
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID441142
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419520675
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID30538
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID411181230
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426146645
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP81800
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID378
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458394811
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCE2RVI8
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID557248
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419499395
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426229348
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID157704013
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP00974
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3866
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCF1SMI0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ05700
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID20517737
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ59149
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9ESD1
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID488746
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458032210
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP28293
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID18760746
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID56538
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9ES87
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID11012
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID456144919
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID452361971
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6GV19
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12734
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID395837
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP09237
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID239
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1991
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ05205
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7937
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP35051
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID409982724
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID21898
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID19143
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP35050
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID290257
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP35049
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID431839318
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID5652
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP09958
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421239125
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419544653
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419500586
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419555088
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID86655555
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP21948
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP00775
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP08311
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID93124
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419516651
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0HJD2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP00764
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419532434
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP23377
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP00761
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9WV82
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0HJC5
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID5045
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100002946
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID162081086
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP19799
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID678603
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6452212
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID414009181
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID25335
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2V898
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9085
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9QX05
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID451509
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415792633
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP81071
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCBAG55035
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP81070
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID448003627
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID136085
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID420228793
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID22061552
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID305265
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCAAH14460
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO00206
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID410068132
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID13035
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9MYW3
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419483213
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419482895
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID416057873
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID41206
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419582727
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458394698
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP84122
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6V115
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393661
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID414002958
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID455012031
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID171548
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID426049
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP17977
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID160712110
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1511
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP23188
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419486041
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6WCD5
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419566294
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID286794
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID750
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID3576
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419537453
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID564
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ10738
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3UP87
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2536
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID32604
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID154074513
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID414244
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8SPE9
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID453652
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP50280
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID243084
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID281536
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8SPE8
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID422600743
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP24664
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415831295
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID30538
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID1476581
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16130295
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO01945

Total number of triples: 255.