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filingDate 2020-02-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2021-03-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_d3181199f2a8653928b4d5e9a216236f
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_78cd885fe95adcae094fdaca8897fabe
publicationDate 2021-03-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10961211-B2
titleOfInvention Isotopically-stabilized tetronimide compounds
abstract Isotopically-stabilized tetronimide compounds comprising one or more deuterium atoms, derivatives, and intermediates, thereof, including methods for their synthesis, pharmaceutical compositions thereof, and methods of using these compounds to interact with target molecules in cell-free samples, cell- and tissue-based assays, animal models, and in a subject are disclosed. One aspect relates to molecules that modulate the expression or catalytic activity of aspartyl (asparaginyl) β-hydroxylase (ASPH) within or on the surface of a cell. Other aspects of the invention relate to use of the molecules disclosed herein to diagnose, ameliorate, or treat cell proliferation disorders and related diseases. Related aspects include uses of the compounds to modulate the activity of viruses, as anti-hyperlipidemia agents, and as agents to ameliorate or treat thrombosis and related cardiovascular and metabolic disorders.
priorityDate 2019-02-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID451638966
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226603258
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID447531973
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5798
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID7474
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393662
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID423563428
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8BSY0
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID154626827
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID154626829
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID795
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID447561522
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16377
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID19098635
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID154626831
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID447561523
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID22087501
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID467868546
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419545310
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID227085755
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID154626832
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453938928
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID447561524
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID53430072
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6995
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393712
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID447574096
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393714
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453950189
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11019101
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226462929

Total number of triples: 1888.