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inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1b1c793981d1946f3ddcea150b6dddce
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publicationDate 2020-06-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10696655-B2
titleOfInvention Therapeutic compounds and uses thereof
abstract The present invention relates to compounds of formula (I) and formula (II): n nand to salts thereof, wherein R 1 -R 4 of formula (I) and R 5 -R 6 of formula (II) have any of the values defined herein, and compositions and uses thereof. The compounds are useful as inhibitors of CBP and/or EP300. Also included are pharmaceutical compositions comprising a compound of formula (I) of formula (II), or a pharmaceutically acceptable salt thereof, and methods of using such compounds and salts in the treatment of various CBP and/or EP300-mediated disorders.
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID294091
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID83722
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24481
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11683
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID161672166
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID430623994
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ865X2
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ865W5
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID397671
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID454887455
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100009081
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Total number of triples: 4846.