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filingDate 2016-09-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2020-06-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f700f8b490d16ac7a23801316b983c08
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publicationDate 2020-06-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10689395-B2
titleOfInvention Tricyclic fused pyridin-2-one derivatives and their use as BRD4 inhibitors
abstract The present disclosure describes heterocyclic compounds of Formula I or, its stereoisomers, pharmaceutically acceptable salts, complexes, hydrates, solvates, tautomers, polymorphs, racemic mixtures, optically active forms and pharmaceutically active derivatives thereof and pharmaceutical compositions containing them as the active ingredient. The present disclosure also describes the synthesis and characterization of aforementioned compounds to exhibit high anticancer activity. The compounds of the present disclosure are useful as medicaments and their use in the manufacture of medicaments for treatment, prevention, or suppression of diseases, and conditions mediated by one or more BET family of bromodomains.
priorityDate 2015-09-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66628417
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100793057
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID126673028
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID333705620
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID126673029
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID333705621
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID126673226
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID126673030
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2794634
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID54694259
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID40467203
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID126673031
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID440710098
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID333705628
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID440710097
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID55717
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID333705630
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID54682893

Total number of triples: 629.