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filingDate 2016-07-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2020-06-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_2c23ef393c2f31432877ec6d6db3c563
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publicationDate 2020-06-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10669234-B2
titleOfInvention Cyanopyrrolidines as dub inhibitors for the treatment of cancer
abstract The present invention relates to novel compounds and method for the manufacture of inhibitors of deubiquitylating enzymes (DUBs). In particular, the invention relates to the inhibition of ubiquitin C-terminal hydrolase L1 (UCHL1) and ubiquitin C-terminal hydrolase 30 or ubiquitin specific peptidase 30 (USP30). The invention further relates to the use of DUB inhibitors in the treatment of cancer and conditions involving mitochondrial dysfunction. Compounds of the invention include compounds having the formula (I) or a pharmaceutically acceptable salt thereof, wherein R 1 , R 2 , R 3 , R 4 , R 5 , R 6 , R 7 , R 8 and R 9 are as defined herein.
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID329722843
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID520170
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID440707356
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Total number of triples: 2245.