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filingDate 2016-09-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2020-05-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5895a6b57c32d89e48da5633214c43b0
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publicationDate 2020-05-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10647675-B2
titleOfInvention Biaryl derivative and medicine containing same
abstract Provided is a compound showing excellent Antifungal activity against Trichophyton fungus, which is a major causative microorganism of superficial mycosis, and high effectiveness on diseases caused by Trichophyton fungi. A biaryl derivative represented by the formula (I) or a salt thereof: n nwherein ring A is an optionally substituted phenyl, or an optionally substituted 5- or 6-membered ring heteroaryl (ring A may be further condensed to form an optionally substituted fused ring); Q is CH 2 , C═O, NH, O, S or the like; X 1 , X 2 and X 3 are CR 1 or N; Y is CH or N; Z is CR 2b or N; R 2a and R 2b are each a hydrogen atom, a halogen atom, an optionally substituted C 1 -C 6 alkyl group, a C 1 -C 6 haloalkyl group or the like; R 2a and R 2b may form, together with carbon atoms bonded thereto, an optionally substituted carbocycle, or an optionally substituted heterocycle.
priorityDate 2015-09-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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Total number of triples: 3378.