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filingDate 2015-12-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2020-04-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_600ced5efeb5f1710bf1cb3e65f63b59
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_7396a9cb6a33bf5d16bf96caaa850da7
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publicationDate 2020-04-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10626140-B2
titleOfInvention Prodrugs of 17β-HSD1-inhibitors
abstract The present invention accordingly provides novel compounds of formula (I) wherein R1, R2, R3 and R4 are as defined in the claims. The invention further relates to their in treatment or prevention of steroid hormone dependent diseases or disorders, such as steroid hormone dependent diseases or disorders requiring the inhibition of the 17β-HSD1 enzyme and/or requiring the lowering of the endogenous estradiol concentration.
priorityDate 2014-12-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5870
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID406041939
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID311183436
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID406041937
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID311183434
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID158987895
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID406041936
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226407967
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID406041935
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399438
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID406041867
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID494003
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID406041866
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135326570
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID406041863
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226519956
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID148387382
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135326567
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ53669
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP70091
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135326566
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135326565
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID158796407
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID9541
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID406042315
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP83456
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID154031900
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135326564
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID87056057
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID161856000
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID406042311
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135326563
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID311183548
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID406041959
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135326578
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394558
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID406041944
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135326577
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID406041943
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID23667301
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135326575
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135326574
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135326573
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID430849294
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP81800
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID403331
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCF2Z4F2
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID449537

Total number of triples: 349.