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grantDate 2020-04-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2020-04-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10617650-B2
titleOfInvention Process for preparing formulations for gastrointestinal-targeted therapies
abstract The present invention provides a process for preparing enterically-coated lyospheres comprising a therapeutic agent comprising: a.) providing lyospheres comprising the therapeutic agent; b.) coating said lyospheres with an enteric polymer coating composition; and c.) isolating said enterically-coated lyospheres. In other embodiments, the invention provides dosage forms comprising a lyosphere comprising an effective amount of a therapeutic agent and an enteric polymer coating. In some embodiments, the therapeutic agent in the process or dosage form is a polypeptide, a protein, a peptide, a lipopeptide, a glycoprotein, a fusion protein, a protein conjugate, a cytokine, an enzyme, an antibody, an oligonucleotide, a vaccine vector, small molecule, a live virus, an inactivated virus, a virus-like particle, a viral protein subunit, an adjuvant, microbiome, a prebiotic, a probiotic, or an ectobiotic. In some embodiments of the present invention, after oral administration the dosage forms containing the enterically-coated lyospheres provide a method of delivering a therapeutic agent to the ileum, ileo-caecal junction, colon or a combination thereof in a subject.
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0KIY3
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID281096
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0KIY2
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393714
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP07321
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0KIY1
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393712
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0KIY0
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID10376
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP04250
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP04249
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID249737
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP04248
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID13856
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0HJQ9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP04247
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID10335
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID126941
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP49672
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2265
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID393558
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399858
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID4151
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID397249
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226492538
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6JV22
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID1496
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID1496
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP32428
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7M424
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID11983
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226402946
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP20856
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226405558
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP30562
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP09965
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226405557
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396047
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396046
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6H8T2

Total number of triples: 345.