http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-10562908-B2

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assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_8c1ee19e6efdf91c1bf88bde9e9845ef
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P29-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D487-04
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D487-04
filingDate 2017-11-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2020-02-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_734672c0624b6446bc6476df5545f86e
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_ccef1a17b8a15e31e898b29837a08987
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_bc17392ca7cb3999c32ec3af595cd211
publicationDate 2020-02-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10562908-B2
titleOfInvention Ortho substituted phenylpyrazolo- and phenylpyrrolo-pyridazine derivatives having multimodal activity against pain
abstract The present invention relates to ortho substituted phenylpyrazolo- and pyrrolo-pyridazine derivatives having dual pharmacological activity towards both the α2δ subunit, in particular the α2δ-1 subunit, of the voltage-gated calcium channel and the μ-opioid receptor, to processes of preparation of such compounds, to pharmaceutical compositions comprising them, and to their use in therapy, in particular for the treatment of pain.
priorityDate 2016-11-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID151851146
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399840
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID386843747
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID134564067
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID454396699
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID139487015
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID386843748
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID139487011
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID70420125
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID386843754
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395100
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID412141703
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID134564064
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID139487013
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11658374
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID21984547
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID417072243
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID386843755
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395130
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID414322096
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID134564066
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6038
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID69804
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID139487018
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453284053
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9221
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID139487019
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID386843752
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9223
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID386843760
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID386843762
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID17935368
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226436555
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID139486955
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID386843756
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9229
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450105094
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419524677
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16722133
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID129196365
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID222
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID386843763
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID139486960
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID386843765
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID412820213
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID139486957
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID386843772
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393660
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID139486958
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID386843773
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226568561
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453757922
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID386843770
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID15182658
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID386843776
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID412824601
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID139486962
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID386843778
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID139486967
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID386843774
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID428235997

Total number of triples: 1006.