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filingDate 2014-12-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2020-01-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10544191-B2
titleOfInvention Methods and compositions for ribosomal synthesis of macrocyclic peptides
abstract Methods and compositions are provided for generating macrocyclic peptides from genetically encoded, ribosomally produced polypeptide precursors. Also provided are nucleic acid molecules, polypeptides, and methods for generating combinatorial libraries of macrocyclic peptides. These methods can be used to produce vast libraries of conformationally constrained peptide ligands as well as facilitate the functional screening of these libraries to identify compound(s) with desired activity properties.
priorityDate 2013-12-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB8D9J3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP19691
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68396207
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA8GIZ1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9MUG5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8Z8F8
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP36354
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP26589
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8ZQX5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6IT78
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7L9L7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP26590
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3AHV1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6D7J7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9ZLJ1
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226581838
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP14325
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ03556
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7M5J8
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7LKT3
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID107844051
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ63VY0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ86134
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7MPI5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8SR10
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ91DS3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA1VRF5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9RTR9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ91QN9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7TUT1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7MFU7
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395653
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2U846
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7NMN1
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395654
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9U6D3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9M2P1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5K2K7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8W4F3
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID1789
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP09459
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7N9S6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2TU51
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237149354
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8X9H8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB1J2C8
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID102577873
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID2209
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID53397917
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP26030
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9JST9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ86523
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP26037
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID4326903
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB6HYN9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8XMP3
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID54023712
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118195882
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ479I3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP21251
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID31310
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396546
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8STF0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6X1D4
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237755418
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2VBN3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO16305
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB1Y0I4
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID4324384
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID236867317
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7T3T2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6X1D8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ66H61
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID272636
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ66DC5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5QXQ2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO76745
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6PI52
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5PCH8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5QVQ6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO62431
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO60041
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID90495
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100533274
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID4932
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID56777065
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID4609
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2K8A4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB5YQM4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA6VCH9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8FU18
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB5XZG7
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID449076581
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP26029
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID2208
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118195790
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID2190
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB6EHL7
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397126
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118195791
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6R520
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8FL25
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226471310
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118195794
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5GWF4
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID2209
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118195792
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118195793
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID326597
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB0KHV8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ89933
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4E6D7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB1X6L3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP15197
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ4FQ23
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9QL89
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP04353
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118195796
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ02KT5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB1XW11
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID448386598
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118195802
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ74DI7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8DC08
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP83456
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9QJT9
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118195803
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118195800
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118195801
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9Y7Y8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9QSP4
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118195774
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9Y105
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID403924
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7W4T0
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID2190
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9WS40
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP60206
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP81800
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6R2R2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7VU94
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID36329
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB1JG85
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP60204
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9WMB5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP41359
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP60205
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB1IY48
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7WGA6
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID4922
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID97541
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA8I1Q0
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118195786
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9PDP1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA1SS83
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ21X72
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA7WNA9
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118195784
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID232811733
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID2875471
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ08823
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO68142
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9943802
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB1LLC4
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16051955
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA7MGQ9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP27305
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ81ZS7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7NX86

Total number of triples: 810.