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filingDate 2017-10-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2020-01-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10544175-B2
titleOfInvention Crystalline fosaprepitant dicyclohexylamine salt and its preparation
abstract Dicyclohexylamine salt of fosaprepitant (fosaprepitant DCHA), a process for preparing fosaprepitant DCHA, and a use of fosaprepitant DCHA in the preparation of pharmaceutically acceptable fosaprepitant dimeglumine with high purity is provided. Fosaprepitant dimeglumine is prepared by treating fosaprepitant DCHA with an acid to form fosaprepitant, followed by adding N-methyl-D-glucamine to fosaprepitant.
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