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grantDate 2020-01-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_eb26b745fc367ef8a3273b412c7a82bc
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publicationDate 2020-01-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10538513-B2
titleOfInvention Pyrazolo and triazolo bicyclic compounds as JAK kinase inhibitors
abstract The invention provides compounds of formula (I): n nor a pharmaceutically-acceptable salt thereof, wherein the variables are defined in the specification, that are inhibitors of JAK kinases, particularly JAK3. The invention also provides crystalline forms, pharmaceutical compositions comprising such compounds, methods of using such compounds to treat gastrointestinal and other inflammatory diseases, and processes and intermediates useful for preparing such compounds.
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID381547944
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID381547943
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP41683
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO62641
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID451934
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID381547942
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID68888
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397282
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6335613
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397281
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226604612
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID23523
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID571383
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100101579
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP51748
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID381536162
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID18644465
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP51747
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118270628
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP41693
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID157773623
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP51745
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID492350
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP41687
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP51744
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395359
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397126
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP41522
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID381536155
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6JV22
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100004988
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID444036
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395352
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID228279576
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID381536153
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226419990
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID81531
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID381536161
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID381536159
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID234513337
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID59605306
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID381536158
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ04745
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397065
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID381536156
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP19437
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397123
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID743373
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID58438953
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP41324
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2PE78
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID31404
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2PE74
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID368481
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2PE47
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID381536151
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6H8T0
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID23162433
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID381536150
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6H8S9
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID24728098
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396964
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP41159
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2PYN4
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID311989578
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID381536139
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394131

Total number of triples: 1970.