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filingDate 2018-07-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2019-11-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_e7f15de3e9260e9575761550378f2d0d
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publicationDate 2019-11-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10471047-B2
titleOfInvention Method for treating obesity, diabetes, cardiovascular and kidney diseases by regulating GPR30/GPER activity
abstract The current invention is in the field of molecular biology/pharmacology and provides methods of using compounds that modulate the effects of GPR30/GPER for treating obesity and diabetes (preferably agonists) as well as disease states and/or conditions that result from excessive formation of reactive oxygen species (preferably antagonists). These compounds may function as agonists and/or antagonists of the disclosed estrogen receptor and/or modulate the expression/upregulation of nox and nox-associated reactive oxygen species (ROS).
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