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filingDate 2018-12-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2019-08-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2019-08-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10392386-B2
titleOfInvention JAK inhibitors containing a 4-membered heterocyclic amide
abstract The invention provides compounds of formula (I): n nwhich contain a 4-membered heterocyclic amide, where the variables are defined in the specification, or a pharmaceutically-acceptable salt thereof, that are useful as JAK kinase inhibitors. The invention also provides pharmaceutical compositions comprising such compounds, methods of using such compounds to treat respiratory diseases, and processes and intermediates useful for preparing such compounds.
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Total number of triples: 484.