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filingDate 2014-11-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2019-07-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2019-07-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10335366-B2
titleOfInvention Risperidone or paliperidone implant formulation
abstract The present invention is directed to an injectable intramuscular depot composition suitable for forming an in situ solid implant in a body, comprising a drug which is risperidone and/or paliperidone or any pharmaceutically acceptable salt thereof in any combination, a biocompatible copolymer based on lactic and glycolic acid having a monomer ratio of lactic to glycolic acid of about 50:50 and a DMSO solvent, wherein the composition releases the drug with an immediate onset of action and continuously for at least 4 weeks and wherein the composition has a pharmacokinetic profile in vivo that makes it suitable to be administered each 4 weeks or even longer periods.
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