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filingDate 2016-01-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2019-06-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_e901f1b46428540019f17638449a4343
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publicationDate 2019-06-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10307402-B2
titleOfInvention Azabenzimidazole derivatives as agonists of the AMP-activated protein kinase
abstract The present invention relates to compounds of general formula I, wherein the group R 1 , X and Y are defined as in claim 1 , which have valuable pharmacological properties, in particular bind to the AMP-activated protein kinase (AMPK) and modulate its activity. The compounds are suitable for treatment and prevention of diseases which can be influenced by this receptor, such as metabolic diseases, in particular diabetes type 2.
priorityDate 2015-01-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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Total number of triples: 878.