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publicationDate 2019-05-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10287255-B2
titleOfInvention Compounds as histone deacetylase 6 inhibitors and pharmaceutical compositions comprising the same
abstract A compound of formula (I), having histone deacetylase 6 (HDAC6) inhibitory activity, n nwherein X, Q, N, R 1 , R 2 , L, and n are as described, isomers thereof, or pharmaceutically acceptable salts thereof, the use thereof for the preparation of therapeutic medicaments, pharmaceutical compositions comprising the same, a method of treating disease using the composition, and methods for preparing the novel compounds. The novel compounds according to the present invention have histone deacetylase 6 (HDAC6) inhibitory activity, and are effective for the prevention or treatment of HDAC6-associated diseases, including cancer, inflammatory diseases, autoimmune diseases, neurological diseases and neurodegenerative disorders.
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Total number of triples: 3358.