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publicationDate 2019-01-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10173978-B2
titleOfInvention Small molecule androgen receptor inhibitors and methods of use thereof
abstract Small molecule carbazole compounds for use as androgen receptor inhibitors are provided herein. Also provided herein are methods for using the carbazole compounds in treating prostate cancer, including castration-resistant prostate cancer and enzalutamide-resistant prostate cancer. The methods include administering to a subject an effective amount of a compound or composition as described herein.
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100689061
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399921
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID13769
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5XJ10
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB1YD06
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226408624
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226400061
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID22798618
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID448306366
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5364430
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394131
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9MZR1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP41323
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394130
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA4YHA5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO34425
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394128
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9MYV3
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419493516
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID23668834
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3423265
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11776
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA6QP91
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCF6QDM7
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226404050
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ99PS1
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7360
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID4329892
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP40226
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID403045
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID767799
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226404049
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226442256
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA3FFS8
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID728378
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID82153
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226458767
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66602552
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID20317
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID410507621
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO35736
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID2232
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP28773
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226408625
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135274839
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP15692
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419581812
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9XT80
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135274838
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ76BS1
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2375
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC4KHW5
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID31310
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP58839
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135274837
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID463609
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135274836
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO35312
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100766857
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID103023
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID32876
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID232
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP04141
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID126520651
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID24872560
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID395654
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID396526
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0MUT8
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID526279
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394314
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID148124

Total number of triples: 1024.