http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-10155770-B2

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grantDate 2018-12-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b1c401ff1ecc6220b7cf6334b91ab973
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publicationDate 2018-12-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10155770-B2
titleOfInvention Substituted pyrazolopyrimidines and method of use
abstract Compounds of formula (I) n nand pharmaceutically acceptable salts thereof, wherein R 1 , R 2 , R 3 , R 4 , L 1 and G 1 are as defined in the specification, are useful in treating conditions or disorders prevented by or ameliorated by positive allosteric modulation of the γ-aminobutyric acid B (GABA-B) receptor. Methods for making the compounds are described. Also described are pharmaceutical compositions of compounds of formula (I), and methods for using such compounds and compositions.
priorityDate 2015-04-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID853002
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP40130
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122620026
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID319789291
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP14605
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP40137
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122620029
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID319789290
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226614528
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP40135
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122620028
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID319789293
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2758349
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122620031
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID319789292
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP40138
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426248706
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10796753
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122620030
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID319789295
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394128
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122620033
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID319789294
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419532039
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122620032
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID319789297
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394131
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5364430
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3423265
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9VGE8
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122620035
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID319789296
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID227001431
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394130
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421016657
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID8103
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122620034
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID319789300
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9773
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122620037
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID319789299
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8XAP1
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID22798618
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122620036
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12953687
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118100641
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394161
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID21463352
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID423390529
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122620039
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID319789301
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7360
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226404049
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID103023
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID451466370
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID319789304
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122620038
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226763281
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ76L34
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122620041
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID319789303
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID449370593
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID454423580
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ76L33
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122620040
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID319789306
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID433264174
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID18187432
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394200
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID406083
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226404050
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122620043
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID319789305
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226465701
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP40145
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122620042
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID319789308
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419563971
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122620045
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID319789307
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID18462
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP59739
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID319789310
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426209489
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID319789309

Total number of triples: 1017.