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filingDate 2016-06-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2018-10-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_2e388b280ee03275160f6d037630a087
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publicationDate 2018-10-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10112968-B2
titleOfInvention Inhibitors of protein methyltransferase DOT1L and methods of use thereof
abstract The present invention relates to DOT1L inhibitors and methods of identifying, designing, or optimizing them. The present invention also relates to crystals of DOT1L-inhibitor complexes, the crystal structures thereof, and the use of the crystal structures. Also disclosed are pharmaceutical compositions containing these DOT1L inhibitors and methods of treating disorders in which DOT1-mediated protein methylation plays a part, such as cancer and neurological disorders, by administering these compounds and pharmaceutical compositions to subjects in need thereof.
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Total number of triples: 581.