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filingDate 2016-08-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2018-08-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_86146b0bc371459f4a2e9f0e0e79b87b
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publicationDate 2018-08-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10052325-B2
titleOfInvention Heat shock protein binding compounds, compositions, and methods for making and using same
abstract The present subject matter relates to a compound represented by the general formula (I) or (I′) or a pharmacologically acceptable salt thereof; pharmaceutical compositions containing at least one of these compounds; methods of making at least one of these compounds; methods of using at least one of these compounds for treating and/or preventing various cancers and/or proliferation disorders; methods of using at least one of these compounds for monitoring the effectiveness of an anticancer therapy against various cancers. In one embodiment, the subject matter relates to compounds that bind with a level of specificity to heat shock protein 70 (Hsp70). In another embodiment, the subject matter relates to compounds that bind with a level of specificity to inhibit both heat shock protein 70 (Hsp70) and heat shock cognate protein 70 (Hsc70).
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237832256
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9VV43
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7541
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237832252
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419762463
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68381306
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526534
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237832259
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68381311
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526533
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237832277
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419509475
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68381310
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526532
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237832274
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526530
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237832272
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68381316
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID81782
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526537
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237832283
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399996
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237832281
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399995
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24224
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526535
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68381321
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526543
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237832279
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID424691000
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526541
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68381319
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237832300
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID232199494
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526540
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68381318
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237832299
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526539
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237832287
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68381325
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237832285
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID852433
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID527165
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237832748
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226444444
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68381323
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526545
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237832310
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68381330
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66973682
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237832303
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526551
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66973681
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237832301
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526550
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ27571
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526549
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237832752
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68381334
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526548
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237832751
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419814633
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226400163
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526556
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0DTC8
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID424322995
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237832750
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68381332
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66973693
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237832949
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ27ID4
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68381331
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66973692
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237832880
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP22629
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID81822
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68381338
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237832871
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68381337
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526561
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237832838
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68381336
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526560
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68381335
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526559
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66973695
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237832999
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66973694
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID104981
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237832975
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID323922
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68381340
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526564
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68381339
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526563
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526562
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68381345
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526570
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526569
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68381343
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526568
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68381350
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526566
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68381349
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526575
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68381348
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID2538848
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68381347
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID54676860
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68381354
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526579
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID10808
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526576
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526583
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526581
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID424762538
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526580
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68381362
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526587
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID136479235
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID449097368
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226409391
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID574282
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID781
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Total number of triples: 3313.