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publicationDate 2018-07-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10035800-B2
titleOfInvention Substituted 1,4,10-triazadibenzo[cd,f]azulenes, substituted 1,4,5,10-tetraazadibenzo[cd,f]azulenes and substituted 1,4,5,7,10-pentaazadibenzo[cd,f]azulenes as bromodomain inhibitors
abstract The present invention provides for compounds of formula (I) wherein R 1 , R 2 , R 6 , Y 1 , Y 3 , A 1 , A 2 , A 3 and A 4 have any of the values defined in the specification, and pharmaceutically acceptable salts thereof, that are useful as agents in the treatment of diseases and conditions, including inflammatory diseases, cancer, and AIDS. Also provided are pharmaceutical compositions comprising one or more compounds of formula (I).
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID312862960
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID267889
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID420324284
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID432568914
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118863330
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16666
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID312862988
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID428988305
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118863329
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID161067
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5312109
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID312862987
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID428988290
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118863328
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5312108
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID312862986
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID243
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID432733938
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118863335
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226417026
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID312862985
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419562410
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID432733937
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118863334
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID451775394
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226417025
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID312862992
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226414314
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226400003
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118863333
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP42633
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID312862991
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID54145
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID229127305
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66600653
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID422602683
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118863332
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID22462
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID312862990
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID428988521

Total number of triples: 5060.