http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-10035771-B2

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filingDate 2014-05-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2018-07-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2018-07-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-10035771-B2
titleOfInvention Mercaptonicotinic acid compound and preparation method and use thereof
abstract The present invention discloses a class of mercaptonicotinic acid compound and preparation method and use thereof; the general structural formula of the compound is as shown in Formula I. Experiment demonstrates that the mercaptonicotinic acid compound could inhibit activity of botulinum toxin endopeptidase and tetanus toxin endopeptidase in vitro, which has a significant protective effect on botulinum toxin poisoning in mice, and can be used for preparing medicine intended to prevent and/or treat botulism, as well as to prevent botulinum toxin exposure and tetanus.
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Total number of triples: 440.