| abstract |
The invention relates to new annelated carbamoylase heterocycles of interest as potential physiologically active substances (agonists, antagonists and receptor modulators, enzyme inhibitors, oncolytics, antibacterial and antiparasitic agents, etc.), which contains a focused library. compositions comprising as active substance annelated carbamoylaseheterocycles, to methods for their preparation and use. 4] an oxazepane ring annulled with at least one optionally substituted and optionally fused heterocycle Q; , optionally substituted phenyl, optionally substituted aryl, optionally substituted Goethe rocyclyl; Q is pyrrole, pyrazole, imidazole, thiazole, pyrrolidine, indole, benzofuran, 4,5,6,7-tetrahydrobenzothiophene, thieno $ 3.2-b] pyrrole, furo $ 3,2-b] pyrrole, thieno $ 2,3- b] pyrrole, benzimidazole, pyridine, quinoline or 1,2,3,4-tetrahydroisoquinoline cycle. antiparasitic agents, etc.), to a focused library that includes annulus |