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filingDate 2017-01-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2018-06-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_2b410edfc96d25fc79656aa5f2eabfaf
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_230883e8fe89d2074751514cd6e0358d
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publicationDate 2018-06-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber TW-I625334-B
titleOfInvention Novel compound of phosphorus heterocycle and azaphosphorus heterocycle, preparation method thereof and pharmaceutical composition containing same
abstract The invention relates to compounds of formula (I) Its optical isomers and their addition salts with pharmaceutically acceptable acids, where: Ak 1 represents an alkyl chain, X represents-(CH 2 ) m- , -CH (R)-, -N (R )-, -CH 2 -N (R)-, -N (R) -CH 2 -or -CH 2 -N (R) -CH 2- , m and R are as defined in the specification, when X represents-( When CH 2 ) m- , -CH (R)-, -N (R)-, -CH 2 -N (R)-or -N (R) -CH 2- , R 1 and R 2 each represent H, Or when X represents -CH 2 -N (R) -CH 2- , R 1 and R 2 together form a bond, and R 3 represents NH 2 , Cy-NH 2 , Cy-Ak 3 -NH 2 or piperidine-4 -Base, Cy and Ak 3 are as defined in the specification, and R 4 and R 5 (which may be the same or different) each represent H or F. This invention relates to pharmaceuticals.
priorityDate 2016-01-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 399.