http://rdf.ncbi.nlm.nih.gov/pubchem/patent/TW-I226886-B

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filingDate 2000-10-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2005-01-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9860e4e1db402ae306b8d8c0128a92c9
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_4d507394b711c3309437cc8b180dcb2b
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publicationDate 2005-01-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber TW-I226886-B
titleOfInvention Benzamidine derivatives and the pharmacologically acceptable salts thereof, and the pharmaceutical composition thereof for treating or preventing blood coagulation diseases
abstract Benzamidine derivatives of the formula (I), [wherein, R1 is H, a halogen atom, an alkyl group or hydroxyl group; R2 is H, a halogen atom or an alkyl group, R3 is H, an optionally substituted alkyl group, an aralkyl group, an optionally substituted alkanoyl group or an optionally substituted alkylsulfonyl group, R4 and R 5 are the same or different, each represents H, halogen, an optionally substituted alkyl group, an alkoxy group, carboxyl group, an alkoxycarbonyl group or an optionally substituted carbamoyl group, R6 is a substituted pyrrolidinyl group or substituted piperidinyl group] or the pharmaceutically acceptable salts thereof, which have an excellent activated blood coagulation factor X inhibiting effect and useful for treating preventing blood coagulation diseases.
priorityDate 1999-10-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 790.