http://rdf.ncbi.nlm.nih.gov/pubchem/patent/TW-202045166-A

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publicationDate 2020-12-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber TW-202045166-A
titleOfInvention Oral composition, method for manufacturing, and use thereof
abstract An oral composition includes an immediate-release pharmaceutical admixture and an extended-release pharmaceutical admixture. The immediate-release pharmaceutical admixture includes a first portion of an active ingredient and a first portion of a hydrophilic dispersant, in which the active ingredient is substantially insoluble in water. The extended-release pharmaceutical admixture includes a controlled-release material, a second portion of the active ingredient, and a second portion of the hydrophilic dispersant, wherein the second portion of the active ingredient and the second portion of the hydrophilic dispersant are mixed in the controlled-release material, wherein the active ingredient is present as a nanoparticle in the immediate-release pharmaceutical admixture and the extended-release pharmaceutical admixture. The method for manufacturing an oral composition and use of an oral composition for treatment of a symptom or a disease caused by immune response or for treatment of organ rejection are further provided.
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