http://rdf.ncbi.nlm.nih.gov/pubchem/patent/TW-201829421-A
Outgoing Links
Predicate | Object |
---|---|
assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_5b65747ed78f05dd9ebe107b50ce2855 |
classificationCPCAdditional | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P43-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-519 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07B2200-13 |
classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D231-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D519-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P43-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-519 |
classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D519-00 |
filingDate | 2017-12-20-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_530d774a6c0564486567848141889c2c |
publicationDate | 2018-08-16-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber | TW-201829421-A |
titleOfInvention | Method for producing 7H-pyrrolo[2,3-d]pyrimidine derivatives and their cocrystallization |
abstract | The present invention relates to a method for producing a 7H-pyrrolo [2,3-d] pyrimidine derivative used as a Janus kinase (JAK) inhibitor, a co-crystal, a method for producing the co-crystal, and a 7H using the co-crystal -A method for purifying pyrrolo [2,3-d] pyrimidine derivatives. The present invention provides a 3-[(3S, 4R) -3-methyl-6- (7H-pyrrolo [2,3-d] pyrimidin-4-yl) -1,6-diazaspiro [3.4] A method for producing octane-1-yl] -3-oxopropionitrile using, for example, 3-[(3S, 4R) -3-methyl-6- (7H-pyrrolo [2,3-d ] Pyrimidin-4-yl) -1,6-diazaspiro [3.4] octane-1-yl] -3-side propoxynitrile co-crystallized with 3,5-dimethylpyrazole. |
priorityDate | 2016-12-21-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 111.