http://rdf.ncbi.nlm.nih.gov/pubchem/patent/TW-201726131-A

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filingDate 2017-01-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5163f0b69255c8620863d16ec608943d
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publicationDate 2017-08-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber TW-201726131-A
titleOfInvention Macrolide derivative of macrolide lactone immunosuppressant
abstract The object of the present invention is to obtain a preparation which has improved efficacy and safety compared with tacrolimus, and the blood concentration is maintained fixed without individual differences, thereby eliminating the need to control the blood dynamics (valley concentration in the blood). Amount. The present invention relates to a polymer derivative of tacrolimus which is linked to a polyethylene glycol segment of a side chain carboxyl group of a polyaspartic acid derivative and an alcoholic hydroxyl group of tacrolimus.
priorityDate 2016-01-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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