http://rdf.ncbi.nlm.nih.gov/pubchem/patent/TW-201542564-A

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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D495-10
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-407
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filingDate 2014-07-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a2ca16035d1a6a981a3153219c3eb62e
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_e4417c50ea80edc602f1e716ea983061
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http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b0455de2aa8149108426157cd0732654
publicationDate 2015-11-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber TW-201542564-A
titleOfInvention Spiroindoline derivatives and pharmaceutical compositions thereof
abstract The present invention relates to a spiroindoline derivative, a process for the preparation thereof, and a pharmaceutical composition thereof, use thereof for the treatment and/or prevention of a disease, and use thereof for the manufacture of a medicament for treating and/or preventing a disease, These diseases are particularly sexual hormone-related diseases in men and women, especially those selected from the group consisting of endometriosis, uterine fibroids, polycystic ovarian disease, hirsutism, precocious puberty, and gonadotropin-dependent sputum. Tumors (such as prostate cancer, breast and ovarian cancer), gonadotropin pituitary adenomas, sleep apnea, stimulating bowel syndrome, premenstrual syndrome, benign prostatic hypertrophy, contraception and infertility (eg assisted reproductive therapy, such as in vitro labor) Fertilization). This application relates in particular to spiroindoline derivatives as gonadotropin releasing hormone (GnRH) receptor antagonists.
priorityDate 2013-07-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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