| abstract |
The present invention provides an industrially useful novel manufacturing method for an N- porphyrinyl hydrazine derivative having excellent antitumor activity, and a synthetic intermediate thereof.nUsing 2,6-dichloroindole as a raw material, a reaction using 2-(N,N-di-t-butoxycarbonylamino)pyrimidine-5-boronic acid is carried out, and after deprotection and substitution reaction, the objective compound N is obtained. - 啉 嘌呤 嘌呤 嘌呤 derivatives. |