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filingDate 2008-07-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_e69b0486949d628707ce632fcdfd2b8c
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publicationDate 2009-02-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber TW-200906413-A
titleOfInvention Non-basic melanin concentrating hormone receptor-1 antagonists and methods
abstract The present application provides compounds, including all stereoisomers, solvates, prodrugs and pharmaceutically acceptable forms thereof according to Formula I wherein A, R1, R2, R3, R8, and R9 are defined herein. Additionally, the present application provides pharmaceutical compositions containing at least one compound according to Formula I and optionally at least one additional therapeutic agent. Finally, the present application provides methods for treating a patient suffering from an MCHR-1 modulated disease or disorder such as, for example, obesity, diabetes, depression or anxiety by administration of a therapeutically effective dose of a compound according to Formula I.
priorityDate 2007-07-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB8ZS96
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC1CAN3
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA7FGD3
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0BCH1
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6CG57
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419533788
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB5BD44
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC1CIB8
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID914631
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP50595
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4MQT3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6CK57
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP50596
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5WWT7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ98TA8
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100150233
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA4VYR4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA4JH80
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419534378
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID66222139
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ927M8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0ZME2
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419559591
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419534456
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID432284841
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9X1I0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB1KSK4
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100685087
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419521873
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419534469
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8D227
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0A3Q1M1X5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA4VSH4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9X1I8
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419491773
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2YJN9
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419500818
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ749A8
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID58012159
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9HIT1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2KZE4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ4PCS5
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419502484
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5359367
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID410511062
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419522661
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68987
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419549034
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68988
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4843
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO33007
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4QBH8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68989
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP56104
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419559526
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68990
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9A6N3
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419559527
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68991
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4R8N8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68992
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419501289
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ92GY7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC1CPA9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0BMG1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0PM98
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA4QBP4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA7H492
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450006894
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68952
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5X5F4
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419559497
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID58015780
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID3169825
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68953
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100848228
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9XD15
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ97SU1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68954
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68955
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID373802
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4449
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68956
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA8GAV3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01197
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID23937
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68957
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID60605158
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP51642
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01201
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419534484
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID454227566
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO94811
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7U4I1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0PXW7
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419501119
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419534626
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID607641
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID424570892
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB6YRA7
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID3060
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4890
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415993545
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01189
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID31923054
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID40467890
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID12064
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01190
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4RKA2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ706D1
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419534993
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ4QNJ1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP69045
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01191
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID54892
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB6YSN8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB1LBL9
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID31773082
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP69046
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ46IS8
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID2520
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID29593595
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC1CXE5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01192
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID445421
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419535046
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP69047
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB5E6H6
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID167583
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID66671224
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01193
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP69048
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01194
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID6579983
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ46GB9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA4W7F8
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID422601242
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA7MT47
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB9DSX1
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419480172
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2G8V9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA8GT48
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP47417
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ17YK6
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID3885
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6YK33
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4S810
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID159158650
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4RU55
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8DFM1
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID420001197
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4912
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5362129
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9XSW9
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID62816
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5XEB4
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID446156
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5N4R8
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID446157
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID166734
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6332834
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ706D0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9HPA7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ110C6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA8GPC9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB9DYD0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB5EFS1
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID23778370
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID70695641
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ32DF7
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID123195
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ74L69
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA7MP52
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9YA47
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID1182
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0A6V8
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID19246
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ63H69
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB5EXN0

Total number of triples: 2137.