abstract |
THE PRESENT INVENTION RELATES TO ADENOSINE A3 RECEPTOR LIGANDS OF THE GENERAL FORMULA (1); WHITHIN THOSE PREFERABLY ANTAGONISTS; AS WELL AS THEIR SALTS; SOLVATES AND ISOMERS; AND THE PHARMACEUTICAL COMPOSITIONS CONTAININGS THEM; TO THE USE OF THE COMPOUNDS OF THE GENERAL FORMULA (1); AS WELL AS THEIR SALTS; SOLVATES AND ISOMERS; TO THE PREPARATION OF THE COUMPOUNDS OF THE GENERAL FORMULA (1) AND THEIR SALTS; SOLVATES AND ISOMERS; FURTHERMORE TO THE NEW INTERMEDIATES OF THE GENERAL FORMULA (II) AND (III) AND TO THE PREPARATION THEREOF. |